Solid-Phase Synthesis of New Trp(Nps)-Containing Dipeptide Derivatives as TRPV1 Channel Blockers
| Contribuinte(s) |
Universitat de Barcelona |
|---|---|
| Data(s) |
12/03/2014
|
| Resumo |
Trp(Nps)-Lys-NH2 derivatives, bearing alkyl or guanidine groups either at the N-terminus or on the Lys side-chain or at both positions were conveniently prepared on solid-phase and evaluated as TRPV1 channel antagonists. |
| Identificador | |
| Idioma(s) |
eng |
| Publicador |
MDPI Publishing |
| Direitos |
cc-by (c) Pérez de Vega, M.J. et al., 2010 info:eu-repo/semantics/openAccess <a href="http://creativecommons.org/licenses/by/3.0/es">http://creativecommons.org/licenses/by/3.0/es</a> |
| Palavras-Chave | #Síntesi en fase sólida #Canals iònics #Bioquímica #Analgèsics #Ciències de la salut #Proteïnes #Dianes farmacològiques #Solid-phase synthesis #Ion channels #Biochemistry #Analgesics #Medical sciences #Proteins #Drug targeting |
| Tipo |
info:eu-repo/semantics/article info:eu-repo/semantics/publishedVersion |