Transition metal-free Minisci reaction promoted by NCS, and TBHP: acylation of heteroarenes


Autoria(s): Siddaraju, Yogesh; Prabhu, Kandikere Ramaiah
Data(s)

2016

Resumo

A method for acylation for heteroarenes under metal-free conditions has been described using NCS as an additive and TBHP as an oxidant. This method has been successfully employed in acylation of a variety of aldehyde with heteroarenes. The application of the method has been illustrated in synthesizing isoquinoline derived natural products. This strategy provides an efficient, mild and inexpensive method for acylation of heteroarenes. (C) 2015 Elsevier Ltd. All rights reserved.

Formato

application/pdf

Identificador

http://eprints.iisc.ernet.in/53351/1/Tet_72_959_2016.pdf

Siddaraju, Yogesh and Prabhu, Kandikere Ramaiah (2016) Transition metal-free Minisci reaction promoted by NCS, and TBHP: acylation of heteroarenes. In: TETRAHEDRON, 72 (7). pp. 959-967.

Publicador

PERGAMON-ELSEVIER SCIENCE LTD

Relação

http://dx.doi.org/10.1016/j.tet.2015.12.065

http://eprints.iisc.ernet.in/53351/

Palavras-Chave #Organic Chemistry
Tipo

Journal Article

PeerReviewed