Synthesis of substituted 8-aminoquinolines and phenanthrolines through a Povarov approach


Autoria(s): De, Kavita; Legros, Julien; Crousse, Benoit; Chandrasekaran, Srinivasan; Bonnet-Delpona, Daniele
Data(s)

2011

Resumo

The synthesis of 8-aminoquinolines and 1,10-phenanthrolines with substituents in alpha of the nitrogen has been performed through an inverse-demanding aza-Diels-Alder (Povarov reaction) in the fluoroalcohols TFE or HFIP. This path involves simple starting materials: 1,2-phenylenediamines, enol ethers and aldehydes.

Formato

application/pdf

Identificador

http://eprints.iisc.ernet.in/35795/1/Amino.pdf

De, Kavita and Legros, Julien and Crousse, Benoit and Chandrasekaran, Srinivasan and Bonnet-Delpona, Daniele (2011) Synthesis of substituted 8-aminoquinolines and phenanthrolines through a Povarov approach. In: Organic and Biomolecular Chemistry, 9 (2). pp. 347-350.

Publicador

Royal Society of Chemistry

Relação

http://pubs.rsc.org/en/Content/ArticleLanding/2011/OB/c0ob00496k

http://eprints.iisc.ernet.in/35795/

Palavras-Chave #Organic Chemistry
Tipo

Journal Article

PeerReviewed